PRODUCT INFORMATION (Part one)

PHARMACEUTICAL INTERMEDIATES (Part two)


PHARMACEUTICAL INTERMEDIATES ................................................................................

  1. Clenbuterol hcl
    a. 4-aminoacetophenone        min.99%
    b. 4-amino-3,5-dichloroacetophenone
    c. 2-(tert-butylamino)-3,5-dichloro-4-aminoacetophenone hcl        MP: 252-257°C
    d. 1-(amino-3,5-dichlorophenyl)-2-tert-butylaminoethanol        MP:115-122°C
  2. Minoxidil
    2,4-diamino-6-chloropyrimidine min.99%
  3. Clotrimazole
    2-chlorophenyldiphenylchloromethane       MP132-134°C
  4. Piroxicam & meloxicam intermediate
    2-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxylicacidet-hylester-1,1-dioxide MP: 140-143°C
  5. Sulpiride
    a. 2-methoxy benzoic acid
    b. 2-methoxy-5-sulfamoyl benzoic acid
  6. Furosemide
    a. 2,4-dichlorobenzoic acid
    b. 2,4-dichloro-5-sulfamoyl benzoic acid (DSBA)
  7. Imdapamide
    4-chloro-3-sulfamoyl benzoic acid
  8. Bumetanide
    3-nitro-4-chloro-5-sulfamoyl benzoic acid
  9. cefazolin
    a) 1H-terazole acetic acid (TAA)
    b) Methyl mercapto thiadiazole (MMTD)
    c) 1-methyl-5-mercapto terazole (MMT)
    d) Ethyl-2-amino-4-thiazoleacetate (ATA)
  10. Ketoconazole & Miconazole nitrate
    a) 1-acetyl-4-(4-hydroxyphenyl)piperazine         MP: 178-182°C
    b) activity ester
    (cis-[2-(2,4-dichlorophenyl)-2-(1H-imidazol-yl- methyl)-1,3-dioxolane-4-yl]methanol-p-methyl
     sulfonate     MP:117.0-121.0°C
    c) cis-bromo-ester (for itraconazole)         min.98%
        (2RS,4RS)-2-(bromomethyl)-2-(2,4-dichlorophenyl)-1,3-dioxolane -4-methanol benzoate (ester)
    d) imidazole
    e) 1-[2-(2,4-dichlorophenyl)2-hybroxyl]imidazole             MP:134-138°C
    f) 5-chloro-1-methyl-4-nitroimidazole
    g) 2,4-dichloroacetophenone
  11. Ofloxacin & ciprofloxacin
    a) Oxyfluorocarboxylic acid(9,10-difluoro-3-methyl-7-oxo-2,3- Dihydro-7-H-pyrido[1,2,3-de]
    [1,4]ibenzoxazine-6-carboylic acid)         MP: ≥300°C
    b) Q-acid (7-chloro-1-cyclopyl-6-fluoro-1,4-dihydro-4-oxoquinoline-3-carboxylic acid   min.98.5%
    c) 7-chloro-1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxoquinoline- 3-carboxylate        min.98.5%
  12. ß–thymidine and AZT,DDT
     5-methyl-uracil        MP: 320-330°C
  13. Naprosen & Nabumetone
    a.Bromoacrtylyara (2-acetyl-5-bromo-6-methoxy naphthalene        MP: 128°C
    b.ßMethoxy naphthalene (YARA YARA) 2-methoxy-naphthalene
       Methyl-2-naphthyl ether        MP: 72°C
  14. Norfloxacin
    a) 2,4-dichloro-5-fluoroacetophenone        min.99%
    b) 2,4-dichloro-5-fluorobenzoic acid        min.99%
    c) o-fluorobenzoic acid
  15. Chloramphenicol intermediates
     a. para-nitroacetophenone
     b. L-base
     c. S-base
  16. Ketoprofen
     benzophenone-3-propionitrile           min.98%
  17. Dehydration condensing agent
     i. N,N’-dicyclohyxylcarbodiimide (DCC)           MP: 33-35°C
     ii. N,N’-Diisopropylcarbodiimide (DIC)           min.99%
   18. cefatrizin & cefotaxime
     a. (benzothiazol-2-yl)-2-(2-aminothiazol-4-yl)-(z)-2-methoxyimino- thioacetate min.98.5%
     b. ATMIA [2-aminothiazole-4-(methylisoximino acid)]           min.99.0%
     c. DL-phenylglycine           min.98.5%
     d. D(-)phenylglycine           min.98.5%
     e. Potassium ( sodium) salt of D-(-)phenylglycine dance           min.98.5%
   19. carbamazepine
     a. Iminostibene
     b. iminodibenzyl carbonyl chloride
     c. iminostibene carbonyl chloride
     d. 3-chloride-iminodibenzyl
   20. Pantoprazole
     a. 2-chloromethyl-3,4-dimethoxy pyridine hcl
     b. 5-difluoromethoxy-2-mercapto-1-H-benzimidazole

 

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